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List of works by Gabriele Costantino

Cyclopropane derivatives as potential human serine racemase inhibitors: unveiling novel insights into a difficult target

scientific article

Cyclopropane-1,2-dicarboxylic acids as new tools for the biophysical investigation of O-acetylserine sulfhydrylases by fluorimetric methods and saturation transfer difference (STD) NMR.

scientific article published on 31 August 2016

Design and synthesis of trans-2-substituted-cyclopropane-1-carboxylic acids as the first non-natural small molecule inhibitors of O-acetylserine sulfhydrylase

article by Laura Amori et al published 2012 in MedChemComm

Discovering a new class of antifungal agents that selectively inhibits microbial carbonic anhydrases

scientific article published on 01 December 2018

Discovery of Multitarget Agents Active as Broad-Spectrum Antivirals and Correctors of Cystic Fibrosis Transmembrane Conductance Regulator for Associated Pulmonary Diseases

scientific article

Discovery of Multitarget Antivirals Acting on Both the Dengue Virus NS5-NS3 Interaction and the Host Src/Fyn Kinases

scientific article published on 15 June 2015

Discovery of New Potential Anti-Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target-Focused Repurposing Approaches.

scientific article

Rational Design, Synthesis, and Preliminary Structure-Activity Relationships of α-Substituted-2-Phenylcyclopropane Carboxylic Acids as Inhibitors of Salmonella typhimurium O-Acetylserine Sulfhydrylase

scientific article published on 19 February 2016

Target flexibility: an emerging consideration in drug discovery and design

scientific article published on 12 September 2008

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