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List of works by Jean-Marc Plancher

5-hydroxyindole-2-carboxylic acid amides: novel histamine-3 receptor inverse agonists for the treatment of obesity.

scientific article

Adventures in Drug-like Chemistry Space: From Oxetanes to Spiroazetidines and Beyond!

scientific article published on 01 January 2014

Aminothiazole derivatives as neuropeptide Y5 receptor ligands: finding the balance between affinity and physicochemical properties

scientific article published on 01 January 2006

Benzodioxoles: novel cannabinoid-1 receptor inverse agonists for the treatment of obesity

scientific article published on 13 March 2008

Discovery of novel and orally active FXR agonists for the potential treatment of dyslipidemia & diabetes ⬇️

scientific article published on November 12, 2010

Evaluation of tert-butyl isosteres: case studies of physicochemical and pharmacokinetic properties, efficacies, and activities

scientific article published on 28 January 2015

Formation of α-SF5 -Enolate Enables Preparation of 3-SF5 -Quinolin-2-ones, 3-SF5 -Quinolines, and 3-SF5 -Pyridin-2-ones: Evaluation of their Physicochemical Properties

Formation of α-SF5-Enolate Enables Preparation of 3-SF5-Quinolin-2-ones, 3-SF5-Quinolines, and 3-SF5-Pyridin-2-ones: Evaluation of their Physicochemical Properties

scientific article published on 6 January 2016

Gene expression‐based in vivo and in vitro prediction of liver toxicity allows compound selection at an early stage of drug development ⬇️

scientific article published on November 12, 2010

Halogen bonding at the active sites of human cathepsin L and MEK1 kinase: efficient interactions in different environments

scientific article published on September 6, 2011

Identification of an N-oxide pyridine GW4064 analog as a potent FXR agonist

scientific article

Selective naphthalene H(3) receptor inverse agonists with reduced potential to induce phospholipidosis and their quinoline analogs.

scientific article

Stereoselective synthesis of methyl monate C

scientific article published on 01 December 2006

Synthesis and Stability of Oxetane Analogs of Thalidomide and Lenalidomide

scientific article published on 12 August 2013

Systematic Investigation of Halogen Bonding in Protein–Ligand Interactions ⬇️

scientific article published on January 3, 2011

The Histamine H3 Receptor as a Therapeutic Drug Target for Metabolic Disorders: Status, Challenges and Opportunities ⬇️

scientific article published on January 1, 2011

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