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List of works by W. Armand Guiguemde

(+)-SJ733, a clinical candidate for malaria that acts through ATP4 to induce rapid host-mediated clearance of Plasmodium.

scientific article

An all-purpose antimalarial drug target

scientific article published on June 2012

Chemical genetics of Plasmodium falciparum

scientific article (publication date: 20 May 2010)

Dihydroquinazolinone inhibitors of proliferation of blood and liver stage malaria parasites

scientific article

Discovery of novel antimalarial compounds enabled by QSAR-based virtual screening

scientific article published on 23 January 2013

Discovery of novel, orally bioavailable, antileishmanial compounds using phenotypic screening.

scientific article published on 29 December 2017

Evaluation of Diarylureas for Activity Against Plasmodium falciparum.

scientific article

Evaluation of histone deacetylase inhibitors (HDACi) as therapeutic leads for human African trypanosomiasis (HAT).

scientific article published on 2 January 2015

Global phenotypic screening for antimalarials

scientific article

Identification of Selective Inhibitors of the Plasmodium falciparum Hexose Transporter PfHT by Screening Focused Libraries of Anti-Malarial Compounds

scientific article

Lead optimization of 3-carboxyl-4(1H)-quinolones to deliver orally bioavailable antimalarials

scientific article

Lead optimization of antimalarial propafenone analogues.

scientific article published on 29 June 2012

Open Source Drug Discovery with the Malaria Box Compound Collection for Neglected Diseases and Beyond

scientific article (publication date: July 2016)

Optimization of propafenone analogues as antimalarial leads

scientific article published on 10 October 2011

PfCHA is a mitochondrial divalent cation/H+ antiporter in Plasmodium falciparum

scientific article (publication date: June 2010)

Potent Plasmodium falciparum gametocytocidal activity of diaminonaphthoquinones, lead antimalarial chemotypes identified in an antimalarial compound screen.

scientific article

Synthesis and evaluation of 7-substituted 4-aminoquinoline analogues for antimalarial activity

scientific article published on 26 September 2011

Synthesis and structure-activity relationships of antimalarial 4-oxo-3-carboxyl quinolones.

scientific article published on 11 February 2010

Treatment of murine cerebral malaria by artemisone in combination with conventional antimalarial drugs: antiplasmodial effects and immune responses.

scientific article

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