Search filters

List of works by Mariangela Urbano

Antagonists of the kappa opioid receptor

scientific article (publication date: May 2014)

C-H activation reactions as useful tools for medicinal chemists

scientific article

Design and Synthesis of a Novel and Selective Kappa Opioid Receptor (KOR) Antagonist (BTRX-335140)

scientific article published on 13 February 2019

Design, synthesis and SAR analysis of novel potent and selective small molecule antagonists of NPBWR1 (GPR7) ⬇️

scientific article published on October 2, 2012

Design, synthesis and SAR analysis of novel selective sigma1 ligands (Part 2).

scientific article published on 21 December 2009

Design, synthesis, and SAR analysis of novel selective sigma1 ligands.

scientific article

Discovery, design and synthesis of a selective S1P(3) receptor allosteric agonist

scientific article

Discovery, design and synthesis of novel potent and selective sphingosine-1-phosphate 4 receptor (S1P₄-R) agonists

scientific article

Discovery, design and synthesis of the first reported potent and selective sphingosine-1-phosphate 4 (S1P4) receptor antagonists

scientific article

Discovery, synthesis and SAR analysis of novel selective small molecule S1P4-R agonists based on a (2Z,5Z)-5-((pyrrol-3-yl)methylene)-3-alkyl-2-(alkylimino)thiazolidin-4-one chemotype ⬇️

scientific article published on September 20, 2011

Enantioselective chromatography and absolute configuration of N,N-dimethyl-3-(naphthalen-2-yl)-butan-1-amines: potential sigma1 ligands

scientific article published in May 2006

Highly diastereoselective synthesis of enantiopure naphthylaminoalcohols with analgesic properties

scientific article published on 01 November 2006

Identification of a Novel Agonist of the Sphingosine 1-phosphate Receptor 4 (S1P4)

Identification of a potent and selective σ₁ receptor agonist potentiating NGF-induced neurite outgrowth in PC12 cells

scientific article published on 14 September 2011

Microwave-assisted extraction of coumarin and related compounds from Melilotus officinalis (L.) Pallas as an alternative to Soxhlet and ultrasound-assisted extraction.

scientific article published in September 2006

Modulators of the Sphingosine 1-phosphate receptor 1.

scientific article published on 29 September 2013

Optimization and Characterization of a Second Antagonist for G-protein Coupled Receptor 7 (GPR7)

Optimization and Characterization of an Antagonist for G-Protein Coupled Receptor 7 (GPR7) ⬇️

scientific article published on July 27, 2012

Probe Development Efforts to Identify Novel Agonists of the Sphingosine 1-phosphate Receptor 4 (S1P4) ⬇️

scientific article published on July 27, 2012

SAR analysis of innovative selective small molecule antagonists of sphingosine-1-phosphate 4 (S1P4) receptor ⬇️

scientific article published on July 13, 2011

SAR analysis of novel non-peptidic NPBWR1 (GPR7) antagonists

scientific article published on 20 December 2012

Sphingosine 1-phosphate receptor 1 agonists: a patent review (2013-2015).

scientific article published on 7 March 2016

Sphingosine 1-phosphate receptor agonists: a patent review (2010-2012)

scientific article

Substituted benzylaminoalkylindoles with preference for the sigma2 binding site.

scientific article published on 26 September 2007

Paulina is supported by:

About Paulina

Help