List of works - Andrea Schweinitz

4-amidinobenzylamine-based inhibitors of urokinase

scientific article published on 01 February 2002

Correlating structure and ligand affinity in drug discovery: a cautionary tale involving second shell residues

scientific article

Crystals of urokinase type plasminogen activator complexes reveal the binding mode of peptidomimetic inhibitors

scientific article (publication date: 18 April 2003)

Design of novel and selective inhibitors of urokinase-type plasminogen activator with improved pharmacokinetic properties for use as antimetastatic agents

scientific article

From selective substrate analogue factor Xa inhibitors to dual inhibitors of thrombin and factor Xa. Part 3

scientific article published on 06 April 2007

Highly potent and selective substrate analogue factor Xa inhibitors containing D-homophenylalanine analogues as P3 residue: part 2

scientific article published on 01 July 2007

Hydrophobic alkyl chains substituted to the 8-position of cyclic nucleotides enhance activation of CNG and HCN channels by an intricate enthalpy - entropy compensation

scientific article published in Scientific Reports

In vitro inhibition of matriptase prevents invasive growth of cell lines of prostate and colon carcinoma

scientific article published on October 2005

Incorporation of neutral C-terminal residues in 3-amidinophenylalanine-derived matriptase inhibitors

scientific article published on 14 February 2009

Increase of anti-metastatic efficacy by selectivity- but not affinity-optimization of synthetic serine protease inhibitors

scientific article published on October 2003

Modification of the N-terminal sulfonyl residue in 3-amidinophenylalanine-based matriptase inhibitors

scientific article published on 13 November 2008

New substrate analogue inhibitors of factor Xa containing 4-amidinobenzylamide as P1 residue: part 1

scientific article published on 01 July 2006

Novel Fluorescent Cyclic Nucleotide Derivatives to Study CNG and HCN Channel Function

scientific article published on 10 May 2019

Relating ligand binding to activation gating in P2X2 receptors using a novel fluorescent ATP derivative

scientific article published on 28 December 2019

Secondary amides of sulfonylated 3-amidinophenylalanine. New potent and selective inhibitors of matriptase

scientific article published on 01 July 2006

Structure-activity relationships of new NAPAP-analogs.

scientific article published in April 2002

Tick-borne Diseases (Borreliosis, Anaplasmosis, Babesiosis) in German and Austrian Dogs: Status quo and Review of Distribution, Transmission, Clinical Findings, Diagnostics and Prophylaxis

scientific article published on August 2015

Use of IHC and newly designed matriptase inhibitors to elucidate the role of matriptase in pancreatic ductal adenocarcinoma

scientific article

List of works by Andrea Schweinitz

4-amidinobenzylamine-based inhibitors of urokinase

Correlating structure and ligand affinity in drug discovery: a cautionary tale involving second shell residues

Crystals of urokinase type plasminogen activator complexes reveal the binding mode of peptidomimetic inhibitors

Design of novel and selective inhibitors of urokinase-type plasminogen activator with improved pharmacokinetic properties for use as antimetastatic agents

From selective substrate analogue factor Xa inhibitors to dual inhibitors of thrombin and factor Xa. Part 3

Highly potent and selective substrate analogue factor Xa inhibitors containing D-homophenylalanine analogues as P3 residue: part 2

Hydrophobic alkyl chains substituted to the 8-position of cyclic nucleotides enhance activation of CNG and HCN channels by an intricate enthalpy - entropy compensation

In vitro inhibition of matriptase prevents invasive growth of cell lines of prostate and colon carcinoma

Incorporation of neutral C-terminal residues in 3-amidinophenylalanine-derived matriptase inhibitors

Increase of anti-metastatic efficacy by selectivity- but not affinity-optimization of synthetic serine protease inhibitors

Modification of the N-terminal sulfonyl residue in 3-amidinophenylalanine-based matriptase inhibitors

New substrate analogue inhibitors of factor Xa containing 4-amidinobenzylamide as P1 residue: part 1

Novel Fluorescent Cyclic Nucleotide Derivatives to Study CNG and HCN Channel Function

Relating ligand binding to activation gating in P2X2 receptors using a novel fluorescent ATP derivative

Secondary amides of sulfonylated 3-amidinophenylalanine. New potent and selective inhibitors of matriptase

Structure-activity relationships of new NAPAP-analogs.

Tick-borne Diseases (Borreliosis, Anaplasmosis, Babesiosis) in German and Austrian Dogs: Status quo and Review of Distribution, Transmission, Clinical Findings, Diagnostics and Prophylaxis

Use of IHC and newly designed matriptase inhibitors to elucidate the role of matriptase in pancreatic ductal adenocarcinoma