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List of works by David H. Coy

(D-Phe12) bombesin and substance P analogues function as central bombesin receptor antagonists

scientific article published in January 1988

A Peptide Inhibitor of Luteinizing Hormone-Releasing Hormone (LH-RH) ⬇️

scientific article published on 01 August 1973

A comparison of the effects of human and ovine corticotropin-releasing hormone on the pituitary-adrenal axis

scientific article published on 01 February 1995

A conjugate of camptothecin and a somatostatin analog against prostate cancer cell invasion via a possible signaling pathway involving PI3K/Akt, alphaVbeta3/alphaVbeta5 and MMP-2/-9.

scientific article published on 27 April 2006

A multi-tyrosinated sst1/2 receptor preferring somatostatin agonist inhibits reflex and immune-mediated secretion in the guinea pig colon

scientific article published in June 2003

A structure-function study of PACAP using conformationally restricted analogs: Identification of PAC1 receptor-selective PACAP agonists

scientific article published on 16 February 2015

Abilities of 3,4-diarylfuran-2-one analogs of combretastatin A-4 to inhibit both proliferation of tumor cell lines and growth of relevant tumors in nude mice.

scientific article published on January 2004

Absence of LH-RH binding sites in corpora lutea from rhesus monkeys (Macacca mulatta)

scientific article published on 01 July 1981

Activity of VIP, somatostatin and other peptides in the mouse vas deferens assay

scientific article published in November 1978

Adenohypophyseal response to hypophysiotropic hormones in male obese Zucker rats

scientific article published in October 1985

Administration of agonistic and antagonistic analogues of LH-RH induce anovulation in Macaca fasicularis

scientific article published on June 1983

Administration of human pancreatic growth hormone-releasing factor (GRF) analogs enhances responsiveness of cultured rat pituitary cells to GRF ⬇️

scientific article published on October 15, 1984

Adrenomedullin Does Not Inhibit Human Platelet Aggregation

scientific article published on 01 July 1998

Adrenomedullin, amylin, calcitonin gene-related peptide and their fragments are potent inhibitors of gastric acid secretion in rats ⬇️

scientific article published on 01 October 1997

An Analog of Enkephalin Having Prolonged Opiate-Like Effects in Vivo ⬇️

scientific article published on April 1, 1977

An adjustable release rate linking strategy for cytotoxin-peptide conjugates

scientific article

An extremely sensitive in vitro model for elucidating structure-activity relationships of growth hormone-releasing factor analogs

scientific article published in January 1985

An in Vivo Assay for Anti-LH-RH and Anti-FSH-RH Activity of Inhibitory Analogues of LH-RH∗ ⬇️

scientific article published on May 1, 1975

An in vivo model for testing inhibition of arginine-induced insulin and glucagon release by somatostatin analogs ⬇️

scientific article published on December 1, 1977

Analogs of luteinizing hormone-releasing hormone containing derivatives of phenylalanine in place of tyrosine ⬇️

scientific article published on July 1, 1973

Analogs of luteinizing hormone-releasing hormone with increased biological activity produced by D-amino acid substitutions in position 6 ⬇️

scientific article published on March 1, 1976

Analogues of growth hormone-releasing factor (1-29) amide containing the reduced peptide bond isostere in the N-terminal region

scientific article published in July 1990

Analysis of cardiovascular and pulmonary responses to endothelin-1 and endothelin-3 in the anesthetized cat.

scientific article published in June 1990

Analysis of responses to hAmylin, hCGRP, and hADM in isolated resistance arteries from the mesenteric vascular bed of the rat.

scientific article published in September 2001

Antagonism of ethanol induced sleep-time by alpha-msh, MSH/ACTH4-10 and naloxone

scientific article published on 01 January 1980

Antagonistic activity of analogs of luteinizing hormone-releasing hormone (LH-RH) in vitro

scientific article published in August 1976

Antagonistic analogs of luteinizing hormone-releasing hormone are mast cell secretagogues

scientific article

Antisense peptide nucleic acids conjugated to somatostatin analogs and targeted at the n-myc oncogene display enhanced cytotoxity to human neuroblastoma IMR32 cells expressing somatostatin receptors

scientific article

Application of human pancreatic carcinoid BON cells for receptor-targeted drug development ⬇️

scientific article published on November 18, 2010

Attempts to induce ovulation in amenorrheic patients using D-Ala-6-LH-RH propylamide

scientific article published on January 1979

Autoradiographic localization of neuromedin B binding sites in rat brain

scientific article published in October 1990

Behavioral effects after systemic injection of opiate peptides

scientific article published on January 1980

Behavioral effects of D-Ala2-beta-endorphin in squirrel monkeys

scientific article published on November 1978

Biological studies with enkephalins and endorphins and their analogs

scientific article published on January 1, 1978

Blockade of LH Release and Ovulation in the Rabbit with Inhibitory Analogues of Luteinizing Hormone Releasing Hormone1 ⬇️

scientific article published on June 1, 1977

Blood-brain barrier, half-time disappearance, and brain distribution for labeled enkephalin and a potent analog ⬇️

scientific article published on November 1, 1976

Bombesin receptor antagonists differentiate receptor subtypes in rat brain

scientific article

Brain β-endorphin-like immunoreactivity in adult rats given β-endorphin neonatally ⬇️

scientific article published on December 1, 1981

Breakdown of enkephalin and endorphin analogs by brain extracts ⬇️

scientific article published on November 1, 1977

CNS effects of peripherally administered brain peptides

scientific article

CNS effects of somatostatin

scientific article published on September 1978

Camptothecin-somatostatin conjugates inhibit the growth of small cell lung cancer cells

scientific article published on 9 April 2005

Characterization of binding sites for N-Tyr-MIF-1 (Tyr-Pro-Leu-Gly-NH2) in rat brain

scientific article

Characterization of bombesin receptors using a novel, potent, radiolabeled antagonist that distinguishes bombesin receptor subtypes ⬇️

scientific article published on May 1, 1993

Characterization of putative GRP- and NMB-receptor antagonist's interaction with human receptors.

scientific article published on 20 May 2009

Chimeric galanin analogs that function as antagonists in the CNS are full agonists in gastrointestinal smooth muscle ⬇️

scientific article published on August 1, 1993

Clinical comparison of natural LH-RH, synthetic LH-RH, and two analogues of LH-RH

scientific article published on 01 May 1974

Cloned somatostatin receptors: identification of subtype-selective peptides and demonstration of high affinity binding of linear peptides

scientific article published on June 1993

Comparative effects of adrenomedullin, an adrenomedullin analog, and CGRP in the pulmonary vascular bed of the cat and rat

scientific article published on 01 January 1995

Comparative pharmacology of bombesin receptor subtype-3, nonpeptide agonist MK-5046, a universal peptide agonist, and peptide antagonist Bantag-1 for human bombesin receptors

scientific article published on 26 July 2013

Comparison of long-acting analogues of luteinizing hormone releasing hormone in man ⬇️

scientific article published on April 1, 1979

Comparison of methionine-enkephalin and morphine in the stimulation of gastric acid secretion in the dog

scientific article published on February 1, 1980

Comparison of prolonged in vivo inhibitory activity of several potent bombesin (BN) antagonists on BN-stimulated amylase secretion in the rat ⬇️

scientific article published on July 1, 1991

Comparison of responses to adrenomedullin and calcitonin gene-related peptide in the feline erection model ⬇️

scientific article published on September 1, 1997

Comparison of the Distribution of Dynorphin Systems and Enkephalin Systems in Brain ⬇️

scientific article published on December 10, 1982

Comparison of the anti-LH/FSH-RH and anti-ovulatory activities of (D-Phe2, D-Leu6)-LH-RH and (D-Phe2, D-Ala6)-LH-RH

scientific article published on 01 January 1976

Comparison of the effect of somatostatin on gastrointestinal function in the conscious and anaesthetized cat and on the isolated cat pancreas ⬇️

scientific article published on July 1, 1977

Comparison of the peptide structural requirements for high affinity interaction with bombesin receptors.

scientific article published in December 1995

Content of beta-LPH and its fragments (including endorphins) in anterior and intermediate lobes of the bovine pituitary gland

scientific article

Correlation Between Luteinizing Hormone Responses to Luteinizing Hormone-Releasing Hormone (LH-RH) And to d-Leu-6-LH-RH-Ethylamide in Patients with Hypothalamo-Pituitary Disease ⬇️

scientific article published on October 1, 1976

Correlation between in vivo inhibition of gonadotropin release induced by LH-RH and the blockade of ovulation by synthetic analogues of LH-RH

scientific article published on January 1, 1978

Corticotrophin releasing factor: responses in normal subjects and patients with disorders of the hypothalamus and pituitary

scientific article published on January 1984

Corticotropin-Releasing Factor Stimulates Secretion of Melanocyte-Stimulating Hormone from the Rat Pituitary ⬇️

scientific article published on July 2, 1982

Corticotropin-releasing factor stimulates accumulation of adenosine 3', 5'-monophosphate in rat pituitary corticotrophs

scientific article published in May 1982

Cranial irradiation for cerebral and nasopharyngeal tumours in children: evidence for the production of a hypothalamic defect in growth hormone release

scientific article published in January 1986

Cyclic analogs of luteinizing hormone-releasing hormone with significant biological activities ⬇️

scientific article published on September 1, 1978

D-Ala2,F5Phe4-dynorphin amide, an opiate with analgesic and toxic properties

scientific article published on March 1, 1992

D-Ala6, Des-Gly-NH210-LH-RH-Ethylamide: A New Analogue with Unusually High LH-RH/FSH-RH Activity ⬇️

scientific article published on 01 October 1974

DSIP reduces amphetamine-induced hyperthermia in mice

scientific article published in August 1984

DSIP-like immunoreactivity in the developing rat brain

scientific article published in December 1981

Degradation of delta sleep inducing peptide (DSIP) and its analogs by brain extracts ⬇️

scientific article published on November 1, 1977

Delta sleep-inducing peptide (DSIP)-like material is absorbed by the gastrointestinal tract of the neonatal rat.

scientific article published in October 1983

Delta sleep-inducing peptide crosses the blood-brain-barrier in dogs: some correlations with protein binding

scientific article

Delta-sleep-inducing peptide reduces CRF-induced corticosterone release

scientific article published in October 1985

Desmethionine alkylamide bombesin analogs: a new class of bombesin receptor antagonists with potent antisecretory activity in pancreatic acini and antimitotic activity in Swiss 3T3 cells ⬇️

scientific article published on January 23, 1990

Development of a potent bombesin receptor antagonist with prolonged in vivo inhibitory activity on bombesin-stimulated amylase and protein release in the rat ⬇️

scientific article published on July 1, 1992

Development of bombesin analogs with conformationally restricted amino acid substitutions with enhanced selectivity for the orphan receptor human bombesin receptor subtype 3.

scientific article published on 21 April 2004

Development of high affinity camptothecin-bombesin conjugates that have targeted cytotoxicity for bombesin receptor-containing tumor cells

scientific article published on 11 March 2004

Development of simplified vasoactive intestinal peptide analogs with receptor selectivity and stability for human vasoactive intestinal peptide/pituitary adenylate cyclase-activating polypeptide receptors

scientific article published on 30 June 2005

Developmental, behavioral, and opiate receptor changes after prenatal or postnatal beta-endorphin, CRF, or Tyr-MIF-1.

scientific article published in January 1985

Differential effects of N-terminal modifications on the biological potencies of growth hormone releasing factor analogues with varying chain lengths

scientific article published in January 1987

Differential penetration of DSIP peptides into rat brain

scientific article

Differentiation of somatostatin receptors involved in inhibition of gastric acid and growth hormone secretion with halogenated Trp8 analogues [proceedings]

scientific article published on December 1, 1978

Direct and indirect inhibition of ovulation in rats by an antagonist of luteinizing hormone-releasing hormone

scientific article published on 01 February 1985

Discovery of a novel class of neuromedin B receptor antagonists, substituted somatostatin analogues.

scientific article published on October 1993

Dissociated effects of somatostatin analogs on arginine-induced insulin, glucagon and growth hormone release in acromegalic patients

scientific article published on 01 October 1983

Distribution of 3H-alpha-MSH in rat brain

scientific article published on January 1, 1976

Distribution of radioactivity in the organs of the rat and mouse after injection of L-(3H)prolyl-L-leucyl-glycinamide

scientific article published on February 1, 1975

Dose response inhibition of the circhoral pulsatile secretion of LH and FSH in rhesus monkeys by the administration of a potent inhibitory analogue of LH-RH ( [N-Ac-D-Trp1, 3, D-p-Cl-Phe2, D-Phe6, D-Ala10]-LH-RH)

scientific article published on 01 July 1983

Dynorphin (1–17): Lack of analgesia but evidence for non-opiate electrophysiological and motor effects ⬇️

scientific article published on October 18, 1982

Effect of D-Trp6-LH-RH on the pituitary-gonadal axis during the luteal phase in the baboon

scientific article published on June 1979

Effect of Somatostatin Analogs on Gastric and Pancreatic Secretion ⬇️

scientific article published on September 1, 1977

Effect of Synthetic Human Pancreatic Growth Hormone-Releasing Factors on Plasma Growth Hormone Concentrations in Lactating Cows ⬇️

scientific article published on 01 December 1984

Effect of Tyr-Pro-Leu-Gly-NH2 on melanotropin-stimulating hormone release in the frog and rat.

scientific article

Effect of a somatostatin analogue on trophic hormone levels in acromegalic patients with elevated hGH after adenomectomy and treatment with bromocriptine

scientific article published on October 1984

Effect of cycloheximide on the LH release induced by a superactive analog of LH-RH

scientific article published on 01 December 1980

Effect of enkephalin and endorphin analogs on receptors in the mouse vas deferens ⬇️

scientific article published on January 1, 1978

Effect of enkephalin and naloxone on gastric acid and serum gastrin and pancreatic polypeptide concentrations in humans

scientific article published on August 1983

Effect of growth hormone release-inhibiting hormone on gastric secretion, mucosal blood flow, and serum gastrin

scientific article published on 01 May 1976

Effect of growth hormone-release inhibiting hormone on hormones stimulating exocrine pancreatic secretion ⬇️

scientific article published on July 1, 1976

Effect of intracerebroventricular administration of beta-/Tyr9/-melanotropin-/9-18/ on rotational behavior induced by substantia nigra lesion in rats

scientific article

Effect of reductive alkylation of D-lysine in position 6 on the histamine-releasing activity of luteinizing hormone-releasing hormone antagonists

scientific article published in April 1987

Effect of somatostatin on gastrointestinal secretions and peptic ulcer production in cats

scientific article

Effect of substitutions in position 12 of bombesin on antagonist activity

scientific article published in May 1989

Effect of the CH2NH and CH2NAc peptide bond isosteres on the antagonistic and histamine releasing activities of a luteinizing hormone-releasing hormone analogue

scientific article published in September 1988

Effects of Administration of a LH-RH Inhibitory Analogue on Stages of the Rat Estrous Cycle ⬇️

scientific article published on October 1, 1978

Effects of H-Phe-Ile-Tyr-His-Ser-Tyr-Lys-OH on passive and active avoidance behavior and on open-field activity of rats

scientific article published on October 1982

Effects of H-Phe-Ile-Tyr-His-Ser-Tyr-Lys-OH on the in vitro uptake and release of radiolabelled dopamine, noradrenaline and serotonin in rat brain hypothalamic slices

scientific article published in May 1984

Effects of a novel bombesin antagonist analogue on bombesin-stimulated gastric acid secretion and growth hormone release in the pentobarbital-anesthetized rat.

scientific article published on January 1989

Effects of an enkephalin analog on complex learning in the rhesus monkey ⬇️

scientific article published on September 1, 1979

Effects of analogs of (pyro)Glu-His-Gly-OH on food consumption and gastric acid secretion in rats

scientific article published on June 1984

Effects of beta-(Tyr9)melanotropin-(9-18) decapeptide on passive and active avoidance behavior and on open-field activity of rats

scientific article published on January 1981

Effects of beta-/Tyr9/melanotropin-/9-18/ on apomorphine-induced stereotyped cage-climbing and on striatal dopamine release in mice. Comparative studies with amphetamine

scientific article

Effects of camptothecin conjugated to a somatostatin analog vector on growth of tumor cell lines in culture and related tumors in rodents

scientific article published on July 2004

Effects of camptothecin on tumor cell proliferation and angiogenesis when coupled to a bombesin analog used as a targeted delivery vector

scientific article published on March 2007

Effects of endorphin and enkephalin analogs on fear habituation in goldfish

scientific article published on July 1, 1978

Effects of in vivo Treatment with an LHRH Antagonist Analog (D-PHE2-D-TRP3-D-PHE6) in the Immature Male Rat1

scientific article published on September 1, 1978

Effects of somatostatin and a somatostatin agonist on diet-induced pancreatitis in mice

scientific article published on November 1985

Elucidation of the vasoactive intestinal peptide pharmacophore for VPAC(2) receptors in human and rat and comparison to the pharmacophore for VPAC(1) receptors

scientific article published in November 2002

Elucidation of vasoactive intestinal peptide pharmacophore for VPAC(1) receptors in human, rat, and guinea pig.

scientific article published in April 2002

Endogenous opiates: 1979(1).

scientific article published on January 1980

Endogenous opiates: 1980 ⬇️

scientific article published on January 1, 1981

Endogenous opiates: 1981 ⬇️

scientific article published on November 1, 1982

Endogenous opiates: Through 1978 ⬇️

scientific article published on January 1, 1979

Enkephalin and a potent analog facilitate maze performance after intraperitoneal administration in rats

scientific article published in December 1976

Enkephalin and other peptides reduce passiveness

scientific article

Entry of DSIP peptides into dog CSF: role of physicochemical and pharmacokinetic parameters

scientific article published in August 1986

Evidence that [125I]N-Tyr-delta sleep-inducing peptide crosses the blood-brain barrier by a non-competitive mechanism

scientific article published in June 1984

Examination of the 1,4-disubstituted azetidinone ring system as a template for combretastatin A-4 conformationally restricted analogue design

scientific article published on May 2004

GI side-effects of a possible therapeutic GRF analogue in monkeys are likely due to VIP receptor agonist activity

scientific article published in July 2001

Galanin-induced relaxation in gastric smooth muscle cells is mediated by cyclic AMP.

scientific article published in January 1994

Gastrointestinal secretory, motor, circulatory, and metabolic effects of prosomatostatin

scientific article

Gonadotropin release during repeated administration of d-Leu6 des Gly10-LH-RH-EA at different stages of the menstrual cycle and in functional amenorrhea

scientific article published on 01 January 1980

Growth hormone release inhibiting hormone: actions on thyrotrophin and prolactin secretion after thyrotrophinreleasing hormone ⬇️

scientific article published on July 12, 1975

HDAC inhibitors suppressed small cell lung cancer cell growth and enhanced the suppressive effects of receptor-targeting cytotoxins via upregulating somatostatin receptor II.

scientific article published on 15 February 2018

High affinity binding of [125I-Tyr11]somatostatin-14 to human small cell lung carcinoma (NCI-H69).

scientific article

Highly active position eight analogues of somatostatin and separation of peptide diastereomers by partition chromatography

scientific article

Highly potent and subtype selective ligands derived by N-methyl scan of a somatostatin antagonist

scientific article published in April 2001

Highly potent cyclic disulfide antagonists of somatostatin

scientific article published in June 1999

Human growth hormone-releasing hormone analogues with much improved in vitro growth hormone-releasing potencies in rat pituitary cells

scientific article published in November 1991

Human pancreatic polypeptide inhibits insulin release in the rat.

scientific article published in July 1981

Hypothalamic Regulatory Hormones ⬇️

scientific article published on January 1, 1978

Hypothalamic hormone interaction in acromegaly ⬇️

scientific article published on September 1, 1975

Identification of a unique ligand which has high affinity for all four bombesin receptor subtypes ⬇️

scientific article published on February 19, 1998

Identification of bombesin receptor subtype-specific ligands: effect of N-methyl scanning, truncation, substitution, and evaluation of putative reported selective ligands.

scientific article published on 30 August 2006

Identification of key amino acids in the gastrin-releasing peptide receptor (GRPR) responsible for high affinity binding of gastrin-releasing peptide (GRP).

scientific article published on 23 December 2004

In VivoInhibition of LH Release by a Synthetic Antagonist of LH-Releasing Hormone (LH-RH)* ⬇️

scientific article published on July 1, 1974

In vitro and in vivo antitumor effects of cytotoxic camptothecin-bombesin conjugates are mediated by specific interaction with cellular bombesin receptors

scientific article published on 9 June 2006

In vitro study of frog (Rana ridibunda Pallas) neurointermediate lobe secretion by use of a simplified perifusion system. III. Effect of neuropeptides on alpha-MSH secretion

scientific article published in November 1983

Inhibition by six somatostatin analogs of plasma growth hormone levels stimulated by thiamylal and morphine in the rat.

scientific article published in January 1976

Inhibition of Release in the Baboon by Inhibitory Analogs of Lutheinizing Hormone Releasing Hormone ⬇️

scientific article published on May 1, 1977

Inhibition of adenosine 3',5'-monophosphate accumulation in anterior pituitary gland in vitro by growth hormone-release inhibiting hormone

scientific article

Inhibition of growth hormone and thyrotropin release by growth hormone-release inhibiting hormone

scientific article

Inhibition of luteinizing hormone release by analogs of luteinizing hormone-releasing hormone (LHRH) in vitro

scientific article published on February 1, 1976

Inhibition of pancreatic secretion by enkephalin and morphine in dogs

scientific article published on May 1, 1978

Inhibition of rat prostate tumor growth by an octapeptide analog of somatostatin

scientific article published on June 1987

Inhibitory Effect of Somatostatin-28 on Pancreatic Polypeptide, Glucagon and Insulin Secretion in Normal Man ⬇️

scientific article published on August 1, 1983

Inhibitory activity of analogues of luteinizing hormone-releasing hormone (LH-RH) in vitro and in vivo

scientific article

Insights into bombesin receptors and ligands: Highlighting recent advances

scientific article

Interaction of galanin fragments with galanin receptors on isolated smooth muscle cells from guinea pig stomach: identification of a novel galanin receptor subtype

scientific article published on 01 January 1995

Interaction of growth hormone-releasing factor (GRF) and 14 GRF analogs with vasoactive intestinal peptide (VIP) receptors of rat pancreas. Discovery of (N-Ac-Tyr1,D-Phe2)-GRF(1-29)-NH2 as a VIP antagonist

scientific article published on 01 June 1985

Inverse relationship between onset and duration of EEG effects of six peripherally administered peptides

scientific article published in December 1981

Investigation of cancer cell lines for peptide receptor-targeted drug development ⬇️

scientific article published on September 1, 2011

Involvement of VPAC1 and VPAC2 receptors in increasing local pancreatic blood flow in anesthetized rats

scientific article published in August 2008

Is the postovulatory release of follicle-stimulating hormone in the rabbit mediated by luteinizing hormone-releasing hormone?

scientific article published in September 1983

Isolation and structure of pro-methionine-enkephalin: Potential enkephalin precursor from porcine hypothalamus

scientific article

Isolation, Structure and Synthesis of a Heptapeptide with In Vitro ACTH-Releasing Activity from Porcine Hypothalamus ⬇️

scientific article published on 01 April 1981

Isolation, structural elucidation and synthesis of a tetradecapeptide with in vitro ACTH-releasing activity corresponding to residues 33-46 of the alpha-chain of porcine hemoglobin

scientific article published on May 1978

Lack of growth hormone-releasing activity of (pyro)Glu-Ser-Gly-NH2.

scientific article published in December 1973

Lanthionine-somatostatin analogs: synthesis, characterization, biological activity, and enzymatic stability studies.

scientific article

Long-acting luteinizing homone-releasing hormone (LH-RH) analogs in the treatment of female infertility

scientific article published on 01 January 1976

Long-term infusion of growth hormone release inhibiting hormone in acromegaly: effects on pituitary and pancreatic hormones.

scientific article

Luteinizing hormone releasing hormone. Solid-phase synthesis of a 5-phenylalanine analog possessing high biological activity.

scientific article published in January 1973

MIF-I and postsynaptic receptor sites for dopamine ⬇️

scientific article published on September 1, 1979

MIF-I's differential actions as an opiate antagonist

scientific article

Metabolism of potent enkephalin analogs (FK 33–824, D-Ala2, pentafluorophenylalanine-4-enkephalinamide and a dimer of D-Ala2-enkephalin) and D-amino acid substituted derivatives of human β-endorphin ⬇️

scientific article published on November 1, 1978

Methionine-Enkephalin Stimulates Gastric Secretion and Gastric Mucosal Blood Flow ⬇️

scientific article published on June 1, 1978

Molecular basis for agonist selectivity and activation of the orphan bombesin receptor subtype 3 receptor.

scientific article published on 15 November 2007

Molecular basis of the selectivity of gastrin-releasing peptide receptor for gastrin-releasing peptide

scientific article published on June 2002

Mu and delta opiate receptors in rat brain are affected by GTP but not by MIF-1.

scientific article published in December 1981

Mu-opiate binding and morphine antagonism by octapeptide analogs of somatostatin

scientific article published in September 1987

N-Methyl scan of somatostatin octapeptide agonists produces interesting effects on receptor subtype specificity

scientific article

Neonatal administration of Met-enkephalin facilitates maze performance of adult rats

scientific article published in December 1980

Neuropeptides and the blood-brain barrier in goldfish

scientific article published on October 1, 1978

New reduced peptide bond substance P agonists and antagonists: effects on smooth muscle contraction ⬇️

scientific article published on October 22, 1991

Nonopiate effects of dynorphin and des-Tyr-dynorphin

scientific article published in December 1982

Novel heptapeptide somatostatin analog displays anti-tumor activity independent of effects on growth hormone secretion

scientific article published on 01 January 1989

Organ distribution of radioactivity and disappearance of radioactivity from plasma after administration of (3H) luteinizing hormone-releasing hormone to mice and rats

scientific article published in January 1974

Parellel inhibition of LH-RH-induced cyclic AMP accumulation and LH and FSH release by LH-RH antagonists in vitro

scientific article published on January 1, 1975

Peptide antagonists of LH-RH: large increases in antiovulatory activities produced by basic D-amino acids in the six position

scientific article published on 01 April 1982

Peptide structural requirements for antagonism differ between the two mammalian bombesin receptor subtypes

scientific article published on October 1995

Peptides readily penetrate the blood-brain barrier: Uptake of peptides by synaptosomes is passive ⬇️

scientific article published on January 1, 1976

Peripheral administration of hypothalamic peptides results in CNS changes

scientific article published on April 1978

Permeability of blood-brain barrier to DSIP peptides

scientific article published in December 1981

Pharmacological characterization of [Leu-13-psi-CH2NH-Leu14]-bombesin as a specific bombesin receptor antagonist on isolated smooth muscle cells

scientific article

Pharmacological characterization of the novel helodermin/VIP receptor present in human SUP-T1 lymphoma cell membranes

scientific article published in September 1989

Pharmacology and intracellular signaling mechanisms of the native human orphan receptor BRS-3 in lung cancer cells ⬇️

scientific article published on October 1, 1998

Pharmacology and selectivity of various natural and synthetic bombesin related peptide agonists for human and rat bombesin receptors differs.

scientific article

Pharmacology of putative selective hBRS-3 receptor agonists for human bombesin receptors (BnR): affinities, potencies and selectivity in multiple native and BnR transfected cells

scientific article

Pituitary adenylate cyclase-activating polypeptide (PACAP) protects against mitoxantrone-induced cardiac injury in mice

scientific article published on 15 July 2017

Pituitary adenylate cyclase-activating polypeptide is a potent broad-spectrum antimicrobial peptide: Structure-activity relationships

scientific article published on 11 April 2018

Pituitary adenylate cyclase-activating polypeptide relaxes rat gastrointestinal smooth muscle

scientific article published on May 1, 1992

Pituitary and Testicular Response to LH-RH and to a Long-Acting Analogue (D-Leu-6-LH-RH-Ethylamide) ⬇️

scientific article published on January 1, 1978

Pituitary response to luteinizing hormone-releasing hormone analog at sea level and high altitudes

scientific article published on 01 January 1982

Plasma gonadotropin response to D-Ala6-LH-RH propylamide

scientific article published on January 1978

Possible non-narcotic component to action of opiate peptides on tonic immobility ⬇️

scientific article published on December 1, 1979

Possible recognition of the GnRH receptor by an antiserum against a peptide encoded by nucleotide sequence complementary to mRNA of a GnRH precursor peptide

scientific article published in November 1986

Potent Antagonists of Somatostatin: Synthesis and Biology ⬇️

scientific article published on March 26, 1998

Potent inhibitory activity of [D-Leu6, Des-Gly-NH2(10)]LHRH ethylamide on LH/hCG and PRL testicular receptor levels in the rat.

scientific article

Presence of highly selective receptors for PACAP (pituitary adenylate cyclase activating peptide) in membranes from the rat pancreatic acinar cell line AR 4-2J.

scientific article published on March 1990

Probing peptide backbone function in bombesin. A reduced peptide bond analogue with potent and specific receptor antagonist activity.

scientific article published on April 1988

Proceedings: Effect of somatostatin on motilin levels and gastric emptying

scientific article published on 01 October 1975

Proceedings: Investigation and treatment of a recurrent vipoma

scientific article

Prolonged Release of LH and FSH and Depletion of Pituitary Gonadotropin Content after Administration of [d-LEU6, desGly-NH210]-LH-RH Ethylamide ⬇️

scientific article published on March 1, 1977

Prolonged inhibition of growth hormone secretion by peripheral injection of bombesin is mediated by somatostatin in the rat

scientific article published on 01 September 1985

Quantitation of somatostatin inhibition of insulin-stimulated gastric acid and pepsin secretion in the cat

scientific article published on June 1, 1978

Radioimmunoassay for GH-Release Inhibiting Hormone ⬇️

scientific article published on March 1, 1975

Radioimmunoassay of DSIP-like material in human blood: possible protein binding

scientific article published in December 1981

Radioimmunoassay of DSIP-like material in rat brain

scientific article published on November 1978

Radioimmunoassay of somatostatin

scientific article published in September 1978

Radioimmunoassayable N-Tyr-MIF-1-like activity in rat brain is increased by pinealectomy

scientific article published in December 1981

Rat melanin concentrating hormone does not modify the release of CRH-41 from rat hypothalamus or ACTH from the anterior pituitary in vitro

scientific article published on October 1990

Recent approaches to fertility control based on derivative of LH-RH.

scientific article published on January 1980

Receptor binding and adenylate cyclase activities of glucagon analogues modified in the N-terminal region

scientific article published in April 1986

Receptor-specific somatostatin analogs: correlations with biological activity

scientific article published on August 1996

Reduced peptide bond pseudopeptide analogues of substance P. A new class of substance P receptor antagonists with enhanced specificity

scientific article published on 01 October 1989

Reduction of distress vocalization in chicks by opiate-like peptides ⬇️

scientific article published on November 1, 1978

Response of human lung tumor xenografts to treatment with a somatostatin analogue (Somatuline).

scientific article published on July 1990

Response to acute administration of pituitary inhibiting hormone, growth hormone and one of its analogues in acromegaly

scientific article published on 01 January 1975

Responses to analogues of growth hormone-releasing hormone in normal subjects, and in growth-hormone deficient children and young adults

scientific article

Role of vagal fibers and bombesin/gastrin-releasing peptide-neurons in distention-induced gastrin release in rats

scientific article published in March 1997

Selective inhibition of glucagon and insulin secretion by somatostatin analogs ⬇️

scientific article published on January 1, 1979

Sensitive radioimmunoassay for somatostatin using N-[125I]-Tyr-somatostatin as labelled antigen ⬇️

scientific article published on January 1, 1979

Serum LH, FSH and testosterone response to the administration of a new LH-RH analog, D-Trp6-LH-RH, in normal men ⬇️

scientific article published on January 1, 1977

Short-chain pseudopeptide bombesin receptor antagonists with enhanced binding affinities for pancreatic acinar and Swiss 3T3 cells display strong antimitotic activity

scientific article published on September 1989

Sleep-wave activity of a delta sleep-inducing peptide analog correlates with its penetrance of the blood-brain barrier

scientific article published in January 1986

Small cell lung cancer bombesin receptors are antagonized by reduced peptide bond analogues.

scientific article

Solid phase synthesis of growth hormone-release inhibiting factor ⬇️

scientific article published on October 15, 1973

Solid-phase synthesis and biological properties of psi [CH2NH] pseudopeptide analogues of a highly potent somatostatin octapeptide

scientific article published in July 1987

Somatostatin analogs which inhibit glucagon and growth hormone more than insulin release

scientific article published in January 1977

Somatostatin receptor subtype 2 mediates inhibition of gastrin and histamine secretion from human, dog, and rat antrum

scientific article published in October 1996

Somatostatin receptor subtypes mediate contractility on human colonic smooth muscle cells.

scientific article published in March 2006

Some analogs of Tyr-MIF-1 affect passive avoidance behavior but not motor activity in rats ⬇️

scientific article published on November 1, 1984

Specific inhibition of rat pancreatic insulin or glucagon release by receptor-selective somatostatin analogs

scientific article published on 01 November 1994

Stereoisomers of luteinizing hormone-releasing hormone ⬇️

scientific article published on July 10, 1974

Stimulation of cyclic AMP accumulation and corticotropin release by synthetic ovine corticotropin-releasing factor in rat anterior pituitary cells: site of glucocorticoid action

scientific article

Stimulation of growth hormone by vasoactive intestinal polypeptide in acromegaly

scientific article published on 01 January 1984

Stimulatory and inhibitory analogs of luteinizing hormone releasing hormone ⬇️

scientific article published on January 15, 1974

Strategies in the design of synthetic agonists and antagonists of growth hormone releasing factor

scientific article published on January 1986

Structural requirements at the N-terminus of urotensin II octapeptides

scientific article published in December 2002

Structural requirements for galanin inhibition of pentagastrin-stimulated gastric acid secretion in conscious rats

scientific article

Structural requirements for the activation of rat anterior pituitary adenylate cyclase by growth hormone-releasing factor (GRF): discovery of (N-Ac-Tyr1, D-Arg2)-GRF(1-29)-NH2 as a GRF antagonist on membranes

scientific article published in November 1985

Structure-NCS activity studies with the enkephalins ⬇️

scientific article published on January 1, 1980

Structure-activity relationships of eighteen somatostatin analogues on gastric secretion ⬇️

scientific article published on April 1, 1978

Structure-activity studies on the N-terminal region of glucagon

scientific article published on March 1984

Structure-activity studies on the N-terminal region of growth hormone releasing factor

scientific article published in February 1985

Studies on the Interaction of Endorphins, Substance P, and Endogenous Somatostatin in Growth Hormone and Prolactin Release in Rats* ⬇️

scientific article published on January 1, 1978

Suppression of gonadotropin release and ovulation in animals by inhibitory analogs of luteinizing hormone-releasing hormone

scientific article published on January 1, 1976

Suppression of postovulatory gonadotropin levels does not affect corpus luteum function in rhesus monkeys

scientific article published on 01 October 1983

Suppression of the positive feedback of estradiol benzoate on gonadotropin secretion by an inhibitory analog of luteinizing hormone-releasing hormone (LRH) in oophorectomized rhesus monkeys: evidence for a necessary synergism between LRH and estroge

scientific article published in August 1983

Suppressive effect of an inhibitory LHRH analog on the gonadotropin response to LHRH in normal women

scientific article published on January 1, 1980

Synthesis and biological activity of position 1 analogs of LH-RH ⬇️

scientific article published on January 1, 1977

Synthesis and biological properties of [Leu-6]-LH-RH and [D-leu-6,desGly-NH210]-LH-RH ethylamide ⬇️

scientific article published on August 19, 1974

Synthesis and biological properties of ovine corticotropin-releasing factor (CRF).

scientific article published in August 1982

Synthesis and opioid activities of stereoisomers and other D-amino acid analogs of methionine-enkephalin

scientific article published in December 1976

Synthetic hypothalamic gonadotropin-releasing hormone (LH-RH) and ovulation: a possibility of "programmed" ovulation to regulate fertility in women (author's transl)

scientific article published on 01 November 1975

Systemic administration of Met-enkephalin, (D-Ala2)-Met-enkephalin, β-endorphin, and (D-Ala2)-β-endorphin: Effects on eating, drinking and activity measures in rats ⬇️

scientific article published on October 1, 1979

Systemic administration of endorphins selectively alters open field behavior of rats ⬇️

scientific article published on May 1, 1978

Temporal changes in FSH and LH concentrations following the administration of a potent LH-RH inhibitory analogue ( [N-Ac-D-Trp1, 3, D-p-Cl-Phe2, D-Phe6, D-Ala10]-LH-RH) to oophorectomized rhesus monkeys

scientific article published on 01 July 1983

The antigenic determinant of the LH-releasing hormone for three different antisera ⬇️

scientific article

The antimicrobial peptides and their potential clinical applications

scientific article published on 15 July 2019

The disappearance, excretion, and metabolism of tritiated prolyl-leucyl-glycinamide in man.

scientific article published in January 1974

The effect of beta-(Tyr9)melanotropin-(9-18) on the active avoidance and open-field behavior on rats pretreated with atropine or propranolol

scientific article published in April 1984

The effect of drug dose and drug exposure time on the binding, internalization, and cytotoxicity of radiolabeled somatostatin analogs

scientific article published on June 2004

The effect of ovine corticotrophin-releasing factor on the hormonal response to insulin-induced hypoglycaemia

scientific article published in February 1989

The half-life, metabolism and excretion of tritiated luteinizing hormone-releasing hormone (LH-RH) in man

scientific article published in October 1973

The interaction between beta-[Tyr9]melanotropin-(9-18), haloperidol and amphetamine in different behavior tests of rats

scientific article published in July 1982

The interaction of growth hormone releasing hormone with other hypothalamic hormones on the release of anterior pituitary hormones

scientific article published in February 1986

The molecular basis for high affinity of a universal ligand for human bombesin receptor (BnR) family members ⬇️

scientific article published on July 22, 2012

The novel VIP-like hypothalamic polypeptide PACAP interacts with high affinity receptors in the human neuroblastoma cell line NB-OK.

scientific article published on July 1990

The pharmacology of endorphin modulation of chick distress vocalization ⬇️

scientific article published on July 1, 1984

The pituitary-adrenal response to CRF-41 is unaltered by intravenous somatostatin in normal subjects

scientific article published in June 1989

The use of a potent stimulatory LHRH analog (D-Trp-6, LHRH) in the induction of ovulation

scientific article published on 01 January 1980

The use of growth hormone-releasing hormone in the diagnosis and treatment of short stature

scientific article

Thyrotrophin and prolactin response to beta-(pyrazolyl-1)-alanine-2-TRH in normal males

scientific article published on 01 February 1981

Tissue distribution of PACAP as determined by RIA: highly abundant in the rat brain and testes

scientific article published in November 1991

Treatment of R-3327 prostate tumors with a somatostatin analogue (somatuline) as adjuvant therapy following surgical castration.

scientific article published in May 1990

Tyr-MIF-1 affects passive avoidance behavior but not motor activity in rats ⬇️

scientific article published on December 1, 1983

Tyr-MIF-1 and MIF-1 are active in the water wheel test for antidepressant drugs

scientific article

Tyr-MIF-1, identified in brain tissue, and its analogs are active in two models of antinociception

scientific article published in December 1985

Unaltered Plasma GH Levels in Acromegalics and Normal Men and Women After Administration of [Pyro]Glu-Ser-Gly-NH2, a Proposed GH-Releasing Hormone* ⬇️

scientific article published on June 1, 1974

Unusual dose-related effect of an endorphin analog in a complex maze

scientific article published in December 1980

VIP attenuation of the severity of experimental pancreatitis is due to VPAC1 receptor-mediated inhibition of cytokine production.

scientific article published in January 2005

Valproic acid induces NET cell growth arrest and enhances tumor suppression of the receptor-targeted peptide-drug conjugate via activating somatostatin receptor type II.

scientific article published on 27 July 2015

Valproic acid suppresses cervical cancer tumor progression possibly via activating Notch1 signaling and enhances receptor-targeted cancer chemotherapeutic via activating somatostatin receptor type II.

scientific article published on 23 February 2013

Vasoactive intestinal peptide reduces oxidative stress in pancreatic acinar cells through the inhibition of NADPH oxidase

scientific article published on 08 September 2011

Vasoactive intestinal peptide-camptothecin conjugates inhibit the proliferation of breast cancer cells

scientific article published on 06 May 2007

[D-Ala2, (F5) Phe4]-dynorphin 1-13-NH2 (DAFPHEDYN): a potent analog of dynorphin 1-13.

scientific article published in September 1987

[Phe4]somatostatin: a potent, selective inhibitor of growth hormone release

scientific article

des-Met carboxyl-terminally modified analogues of bombesin function as potent bombesin receptor antagonists, partial agonists, or agonists

scientific article published on September 1990

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