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A poised fragment library enables rapid synthetic expansion yielding the first reported inhibitors of PHIP(2), an atypical bromodomain† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c5sc03115j.

scientific article published on 22 December 2015

Author/s

author: Patrick M Collins, Romain Talon, John Spencer, Frank von Delft, Paul E. Brennan, Brian D Marsden, Anthony R Bradley, Tobias Krojer

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Publication date
December 22, 2015
- -
Language
English

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