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Lead optimization of a pyrazole sulfonamide series of Trypanosoma brucei N-myristoyltransferase inhibitors: identification and evaluation of CNS penetrant compounds as potential treatments for stage 2 human African trypanosomiasis

scientific article

Author/s

author: Stephen Brand, David A Robinson, Daan van Aalten, Ruth Brenk, Alan Fairlamb, Michael J. Ferguson, Ian H. Gilbert, Laste Stojanovski, Paul G. Wyatt, Kevin D Read, Irene Hallyburton, Neil Richard Norcross, Suzanne Norval, Julie A Frearson, Leah S Torrie, Paul Scullion

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Work details

Publication date
November 20, 2014
- -
Language
English

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