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Receptor residence time trumps drug-likeness and oral bioavailability in determining efficacy of complement C5a antagonists.

scientific article

Author/s

author: Junxian Lim, Mei-Kwan Yau, Weijun Xu, Rink-Jan Lohman, Martin J Stoermer, Matthew J. Sweet, Robert C. Reid, Jacky Y. Suen, David P. Fairlie

Wikidata


Work details

Publication date
April 20, 2016
- -
Language
English

Copyright status